Drug Derivative
Drug derivative
Drug derivatives are derived from parent compounds. They replace or add atoms and groups through chemical reactions to optimize the various properties of the parent compound and reduce side effects. The application of drug derivatives provides a diverse compound library for drug research and development and accelerates the discovery of new drugs. For example, urea derivatives Glibenclamide can prolong the blood sugar-lowering effect of anti-diabetic drugs.
References:
- [1]. Vardanyan RS, et al. Fentanyl-related compounds and derivatives: current status and future prospects for pharmaceutical applications. Future Med Chem. 2014 Mar;6(4):385-412.x
- [2]. Ghosh AK, et al. Urea Derivatives in Modern Drug Discovery and Medicinal Chemistry. J Med Chem. 2020 Mar 26;63(6):2751-2788.x
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Drug Derivative Related Products (4010)
Related Products (4010)
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Anti-virus agent 2
0 ImagesCat. No.: HY-183592Anti-virus agent 2 is an orally active and selective anti-orthopoxvirus (poxvirus) agent, with EC50 values of 6.1 μM and 47.1 μM against VTT-Fluc and MPXV clade IIb, respectively. Anti-virus agent 2 covalently binds to viral A17L protein and mRNA methyltransferase, blocks viral membrane fusion and intracellular biosynthesis, and acts on multiple stages of the viral replication cycle. Anti-virus agent 2 achieves viral inhibition in nude mouse models. Anti-virus agent 2 can be used for the research of orthopoxvirus infections such as monkeypox and smallpox.
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α,α-Trehalose 6-phosphate potassium (Standard)
0 ImagesCat. No.: HY-131368RCAS No.: 136632-28-5Synonyms: Tre6P potassium (Standard)α,α-Trehalose 6-phosphate potassium (Standard) is the analytical standard of α,α-Trehalose 6-phosphate potassium (HY-131368). This product is intended for research and analytical applications. α,α-Trehalose 6-phosphate (Tre6P) potassium is a glucose analogue with potent anti-hyperglcaemic activity. α,α-Trehalose 6-phosphate potassium is rapidly converted to the end product, α,α′-trehalose, through the action of α,α-Trehalose 6-phosphate phosphatase (T6PP).
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β-keto Phentermine hydrochloride
0 ImagesCat. No.: HY-W043333CAS No.: 6946-08-3β-keto Phentermine hydrochloride is a drug derivative.
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Darapladib analog-1
0 ImagesCat. No.: HY-120849CAS No.: 1389264-17-8Darapladib analog-1 (Compound 16) is an O-alkylated Darapladib (HY-10521). Darapladib analog-1 inhibits Lp-PLA2. Darapladib analog-1 can be used in the research of atherosclerosis.
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5-Methoxy EiPT
0 ImagesCat. No.: HY-138162CAS No.: 850032-66-55-Methoxy EiPT is a tryptamine-based designer agent.
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Clopipazan
0 ImagesCat. No.: HY-169128CAS No.: 60085-78-1Clopipazan is a potent antipsychotic agent.
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Oximino Oxamyl-d6
0 ImagesCat. No.: HY-W717863CAS No.: 2734501-51-8Synonyms: Oxamyl oxime-d6Oximino Oxamyl-d6 (Oxamyl oxime-d6) is deuterium labeled Oximino oxamyl. Oximino oxamyl is an active compound.
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OPPD-Q
0 ImagesCat. No.: HY-169493CAS No.: 2952779-34-7OPPD-Q is a p-phenylenediamine-quinone (PPD-Q) and an oxidized derivative of the aromatic amine antioxidant OPPD.
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Antiallergic agent-3
0 ImagesCat. No.: HY-106924ACAS No.: 160665-99-6Antiallergic agent-3 is a derivative of 2-(benzimidazol-2-yl)-1,3-diaminopropane with antiallergic activity.
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Decylplastoquinone
0 ImagesCat. No.: HY-17659CAS No.: 112055-76-2Decylplastoquinone is lipid-soluble derivative of plastoquinone (HY-N11882). Plastoquinone (PQ-9), a potent electron carrier, is an essential component of photosynthesis. Plastoquinone is also a redox sensor that regulates state transitions and gene expression.
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Δ6-Testosterone enanthate
0 ImagesCat. No.: HY-176098CAS No.: 3070439-39-0Δ6-Testosterone enanthate is a synthetic anabolic steroid (AAS), being the Δ6-isomer of testosterone enanthate.
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7(Z),10(Z),13(Z)-Hexadecatrienoic acid methyl ester
0 ImagesCat. No.: HY-168783CAS No.: 77388-16-07(Z),10(Z),13(Z)-Hexadecatrienoic acid methyl ester is a polyunsaturated fatty acid generated during the synthesis of Docosahexaenoic acid-d5 (HY-B2167S).
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4-MAPB hydrochloride
0 ImagesCat. No.: HY-W745320CAS No.: 2742659-53-44-MAPB hydrochloride is a benzofuran compound.
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WAY-620445
0 ImagesCat. No.: HY-149739CAS No.: 728924-73-0WAY-620445 is an active molecule.
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1-Methyl-3-BZP
0 ImagesCat. No.: HY-116201CAS No.: 137539-25-4Synonyms: 3-Benzyl-1-methylpiperazine1-Methyl-3-BZP is a piperazine.
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Glycidyl oleate
0 ImagesCat. No.: HY-W585935CAS No.: 5431-33-4Synonyms: 1-Propanol, 2,3-epoxy-, oleate; Oleic acid glycidyl esterGlycidyl oleate (Oleic acid glycidyl ester) is an ester product.
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8-Oxo-Δ9-THC
0 ImagesCat. No.: HY-179455CAS No.: 37936-78-0Synonyms: 8-Oxo-Δ9-tetrahydrocannabinol; Δ1-Tetrahydrocannabinol-6-one8-Oxo-Δ9-THC is an oxygenated tetrahydrocannabinol that can be found in Cannabis sativa L. variety CHPF-01.
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6-Methoxy DiPT hydrochloride
0 Images6-Methoxy DiPT hydrochloride is structurally categorized as a Tryptamine (HY-B2132).
